Chemical

LDC4297 (LDC044297)

  • Catalog Number : C4049
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General Information

Application Inhibitor
Description  LDC4297 is a novel CDK7 inhibitor (IC50=0.13±0.06 nM for CDK7 versus IC50s between 10 nM and 10,000 nM for all other analyzed CDKs).
Cas NO.  1453834-21-3
Purity  ≥98% 
Molecular Weight 432.52
Formula C23H28N8O
Solubility

DMSO : 86 mg/mL

Ethanol : 86 mg/mL

Water : 27 mg/mL

Target / IC50

CDK7 : 0.13 nM

Alias N/A
Storage

Powder : -20°C for 3 years

 

1 mg

5 mg

10 mg

1 mM

2.3120 mL 11.5602 mL 23.1203 mL
5 mM 0.4624 mL 2.3120 mL 4.6241 mL
10 mM 0.2312 mL 1.1560 mL 2.3120 mL

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