Chemical

Ribociclib (LEE011)

  • Catalog Number : C4043
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General Information

Application Inhibitor
Description 
Ribociclib (LEE011) is an orally available, and highly specific CDK4/6 inhibitor. Phase 3.
Cas NO.  1211441-98-3
Purity  ≥98% 
Molecular Weight 434.54
Formula C23H30N8O
Solubility

DMSO : 7 mg/mL

Ethanol : Insoluble

Water : Insoluble

Target / IC50

CDK4 

CDK6

Alias N/A
Storage

Powder : -20°C for 3 years

 

1 mg

5 mg

10 mg

1 mM

2.3013 mL 11.5064 mL 23.0128 mL
5 mM 0.4603 mL 2.3013 mL 4.6026 mL
10 mM 0.2301 mL 1.1506 mL 2.3013 mL

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