General Information
| Application | Inhibitor |
|---|
| Description | BI-D1870 is a remarkably specific, ATP-competitive inhibitor of RSK isoforms, with IC50 values of 31 nM/24 nM/18 nM/15 nM for RSK1/SK2/SK3/SK4, respectively. |
|---|
| Cas NO. | 501437-28-1 |
|---|
| Purity | ≥99% |
|---|---|
| Molecular Weight | 391.42 |
| Formula | C19H23F2N5O2 |
| Solubility |
DMSO : 10 mM |
|---|
| Target / IC50 |
RSK1 : 31 nM RSK2 : 24 nM RSK3 : 18 nM RSK4 : 15 nM |
|---|
| Alias | N/A |
|---|
| Storage |
Powder : -20°C for 3 years Solvent : -80°C for 6 months |
|---|
|
|
1 mg |
5 mg |
10 mg |
|
|
1 mM |
2.5548 mL | 12.7740 mL | 25.5480 mL | |
| 5 mM | 0.5110 mL | 2.5548 mL | 5.1096 mL | |
| 10 mM | 0.2555 mL | 1.2774 mL | 2.5548 mL | |
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